Cabergoline (that is most famous sold under trade name Cabaser and Dostinex – but there are many others), which is an ergot derivative, is a potent dopamine receptor agonist on D2 receptors. There are studies proving that Cabergoline is directly inhibiting pituitary lactotroph (prolactin) cells. Very often, this product is used in the management of prolactinomas because of its higher affinity for the D2 receptor sites and less severe side effects. This product is known to have only one route of administration – oral, which means that all the products containing Cabergoline should be in form of tablet. The product got popular in the world of bodybuilding because of its ability to offer an “adrenaline rush” and ignoring pains while pushing muscles. But it is mainly used as a prolactin inhibitor.

Below you are going to find all the products containing Cabergoline and you are also going to find a lot of valuable information about this product.

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What is Cabergoline (Cabaser)?

Cabergoline which can be found in many different trade names including Cabaser and Dostinex, is a potent dopamine receptor agonist. Since it is inhibiting prolactin, the current medicine preferred Cabergoline instead of older Bromocriptine because it has a longer half life and less side effects.

The product was discovered in early 1980’s and since 1996 it got FDA approval. The product is a long lasting dopamine D2 receptor agonist. It inhibits the prolactin – a hormone best known to produce female mammals milk, but it has other functions in both males and females.

By using Cabergoline, the prolactin hormone is not being produced so its levels are dropping down. In males, the effect of prolactin is during and after ejaculation. This is the sexual refractory period in which males are losing interest in sex.

What is Cabergoline Used For?

In the medical setting, this substance is used for treatment of different health conditions such as: prolactin producing tumors, parkinson’s disease, cushing’s disease, hyperprolactinemia as well as a myriad of other ailments. But it is best known to be used for tumors and cancers related to high prolactin levels.

However, when this product is used in bodybuilding – it has several ways that can be used. Being a dopamine agonist, there are some sportsmen believing that they can use it to offer an adrenaline rush when is needed during an event or show. This product is believed to improve your motor skills and would make you able to work out a lot much harder than you normally would because you would get pains. With Cabergoline – you should be able to ignore pain and therefore you can push your muscles to the limit.

Anyway, the main reason why bodybuilders are using Cabergoline is because they need it during the cycle when they are running a compound that is increasing levels of prolactin in the body. A good example would be Trenbolone – a famous steroid used by lots of bodybuilders. This steroid will turn into prolactin and if used in high doses, you can get gynecomastia secondary to prolactin levels.

Plus to this, having a too high prolactin levels – this can greatly diminish your sex drive. Cabaer (Cabergoline) can greatly help you to normalize libido even if you’re not using steroids increasing prolactin levels. It can be used even when you are trying some changes on your hormones.

But there’s also another way in which Cabergoline might be used in bodybuilding. That’s in its mechanism of action in which it mimics dopamine that is produced from food intake. In short, it can greatly help those people who are having cravings for some junk/ unhealthy foods such as pizza, ice cream or whatever else that shouldn’t be eaten. By using Cabergoline, the dopamine is released and is acting as a pleasure chemical making you have less cravings. Therefore, it is obvious that this helps with weight loss.

Cabergoline has been discovered to have a close relationship with sex. For example, it was earlier mentioned that prolactin levels is what makes a man lose interest in sex. By using cabergoline – you decrease the prolactin levels and therefore your libido is enhanced. For example, when a man ejaculates, his prolactin levels are spiking up causing him to lose the interest in sex. When supplementing with Cabergoline, your sex drive is recovered quicker.

Cabergoline Dosage | Cabergoline Bodybuilding Administration | Half Life

It was earlier mentioned that Cabergoline has appeared on the market and blown away bromocriptine because it has a much longer half life and much better side effects profile. We would talk about side effects later. As for now Cabergoline has a half life very long of 3 days.

This product is extremely powerful with very long half life. This is the reason why bodybuilders only need to use it 2 times a week and they might use a very low dosage of it and it would be enough to control the prolactin levels. It is recommended to use a dosage only 0.25 mg per dose which means a total dose of 0.5 mg per week.

There are very rare instances when a dose of 0.5 mg per week (taken in 2 different days) won’t be enough. Remember this is a very potent drug and must be taken with big caution.

Cabergoline Side Effects

When using this product abusively it can offer side effects. Most people using it properly won’t experience side effects. Most common side effects from bodybuilders include stomach pains while on Cabergoline.

However, if the product is used at a proper dose and is used with food – this shouldn’t be a problem. Other side effects that are less serious and rarely seen: numbness, nausea, vomiting, dizziness, constipation and some others. But if it’s used before bed with a meal – it should decrease the side effects.

Where To Buy Cabergoline?

Cabergoline that is often sold under trade names – Dostinex, Cabaser or others, is a product that can greatly help if you’re having too high prolactin levels. You can purchase it directly from our website by choosing one of the products you can find above. You are ensured to get the highest quality and lowest possible price on the market.